Ionic liquid-enabled synthesis, cholinesterase inhibitory activity, and molecular docking study of highly functionalized tetrasubstituted pyrrolidines.

TitleIonic liquid-enabled synthesis, cholinesterase inhibitory activity, and molecular docking study of highly functionalized tetrasubstituted pyrrolidines.
Publication TypeJournal Article
Year of Publication2018
AuthorsKumar RSuresh, Almansour AI, Arumugam N, Althomili DMohammed Q, Altaf M, Basiri A, D K, Manohar TSai, S V
JournalBioorg Chem
Volume77
Pagination263-268
Date Published2018 Apr
ISSN1090-2120
Abstract

A small library of novel spiropyrrolidine heterocyclic hybrids has been prepared regioselectively in 1-butyl-3-methylimidazoliumbromide ([bmim]Br) with good to excellent yields using a [3+2] cycloaddition reaction. These synthesized compounds were evaluated as potential agents for treating Alzheimer's disease. Compound 4b showed the most potent activity, with an IC of 7.9 ± 0.25 µM against acetylcholinesterase (AChE). The inhibition mechanisms for the most active compounds on AChE and butyrylcholinesterase (BChE) receptors were elucidated using molecular docking simulations.

DOI10.1016/j.bioorg.2018.01.019
Alternate JournalBioorg. Chem.
PubMed ID29421701

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